2. Characterisation of agonist-receptor interaction. Occupancy, affinity, dose-response curve, potency, efficacy: Revision history

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10 March 2023

  • curprev 15:2215:22, 10 March 2023‎ Nikolas talk contribs‎ 14,650 bytes +14,650‎ Created page with "A quick summary: * Occupancy shows the fraction of the total number of receptors in the tissue that is occupied by the drug. It’s determined by the constant ''p.'' * A drug’s affinity to its receptor is determined by the constant Kd. When Kd is low is the affinity high. A high affinity is always good and has no drawbacks. * Efficacy is a measure of how “effective” the drug is. It measures how large of a cellular response the drug can induce in the tissue, which..." Tag: Visual edit